Search Result "hPXR activators"


Classification of Human Pregnane X Receptor (hPXR) Activators and Non-Activators by Machine Learning Techniques: A Multifaceted Approach

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 19 Issue: 4 Year: 2016 Page: 307-318
Author(s): Vijay Rathod,Vilas Belekar,Prabha Garg,Abhay T. Sangamwar

Evaluation of 170 Xenobiotics as Transactivators of Human Pregnane X Receptor (hPXR) and Correlation to Known CYP3A4 Drug Interactions

Journal: Current Drug Metabolism
Volume: 7 Issue: 4 Year: 2006 Page: 375-388
Author(s): Michael Sinz, Sean Kim, Zhengrong Zhu, Taosheng Chen, Monique Anthony, Kenneth Dickinson, A. D. Rodrigues

Impact of Ritonavir, Atazanavir and Their Combination on the CYP3A4 Induction by Efavirenz in Primary Human Hepatocytes

Journal: Drug Metabolism Letters
Volume: 4 Issue: 1 Year: 2010 Page: 45-50
Author(s): Ganesh M. Mugundu, Niresh Hariparsad, Pankaj B. Desai

Current In Vitro High Throughput Screening Approaches to Assess Nuclear Receptor Activation

Journal: Current Drug Metabolism
Volume: 11 Issue: 9 Year: 2010 Page: 806-814
Author(s): Judy L. Raucy, Jerome M. Lasker

Structure-Activity Relationship of Nuclear Receptor-Ligand Interactions

Journal: Current Topics in Medicinal Chemistry
Volume: 3 Issue: 1 Year: 2003 Page: 1573-1599
Author(s): Holger Greschik, Dino Moras

Counter-Regulatory Role of Bile Acid Activated Receptors in Immunity and Inflammation

Journal: Current Molecular Medicine
Volume: 10 Issue: 6 Year: 2010 Page: 579-595
Author(s): S. Fiorucci, S. Cipriani, A. Mencarelli, B. Renga, E. Distrutti, F. Baldelli

Research Article

Scutellarin Mediates Cytochrome P450 3A4 and 2C19 Expression viaPregnane X Receptor and Constitutive Androstane Receptor

Journal: Current Molecular Pharmacology
Volume: 16 Issue: 6 Year: 2023 Page: 640-653
Author(s):

Review Article

Nociceptin /Orphanin FQ Peptide (NOP) Receptor Modulators: An Update in Structure-Activity Relationships

Journal: Current Medicinal Chemistry
Volume: 25 Issue: 2 Year: 2018 Page: 2353-2384
Author(s): Carlo Mustazza,Stefano Pieretti,Francesca Marzoli

Activation of CAR and PXR by Dietary, Environmental and Occupational Chemicals Alters Drug Metabolism, Intermediary Metabolism, and Cell Proliferation

Journal: Current Pharmacogenomics and Personalized Medicine
Volume: 7 Issue: 2 Year: 2009 Page: 81-105
Author(s): Juan P. Hernandez, Linda C. Mota, William S. Baldwin

New Opportunities for Pregnane X Receptor (PXR) Targeting in Drug Development. Lessons from Enantio- and Species-Specific PXR Ligands Identified from A Discovery Library of Amino Acid Analogues

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 7 Issue: 6 Year: 2007 Page: 617-625
Author(s): Peter Wipf, Haibiao Gong, Jelena M. Janjic, Song Li, Billy W. Day, Wen Xie

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